Temporal Trends in Serious Adverse Events Associated with Oral Antivirals During the COVID-19 Pandemic: Insights from the FAERS Database (2020–2023)

Siby et al., Open Forum Infectious Diseases, doi:10.1093/ofid/ofaf695.1825, Jan 2026
Retrospective 11,547 serious adverse event reports from the FDA database (2020-2023) showing significant safety signals with oral COVID-19 antivirals. Paxlovid showed the strongest signals for drug-drug interactions (ROR: 4.83) and liver injury (ROR: 2.89), while molnupiravir was associated with neurological events (ROR: 2.14) and acute kidney injury (ROR: 1.76), and favipiravir was associated with liver injury and cardiovascular events.
Study covers molnupiravir, paxlovid, and favipiravir.
Siby et al., 11 Jan 2026, retrospective, peer-reviewed, 3 authors, study period January 2020 - December 2023.
Abstract: 1 2 3 1 Faculty of Medicine, Suez University, Suez, Egypt, Suez, As Suways, Egypt 2Faculty of Oral and Dental Medicine, Egyptian Russian University, Badr City, Al Qahirah, Egypt 3Faculty of Medicine, Suez University, Suez, As Suways, Egypt Abstract citation ID: ofaf695.1825 Session: 219. COVID-2019 and Co-Infections Wednesday, October 22, 2025: 12:15 PM Background. The COVID-19 pandemic led to the widespread use of emergency-authorized and repurposed oral antivirals, including remdesivir (initial IV use, later oral analogues), favipiravir, molnupiravir, and nirmatrelvir-ritonavir (Paxlovid). While these agents have played a key role in outpatient COVID-19 management, their real-world safety profiles remain under continuous evaluation. This study aimed to assess the temporal trends and disproportionality of serious adverse events (SAEs) associated with oral antivirals during the pandemic using the U.S. FDA Adverse Event Reporting System (FAERS). 1 2 4 6 9 1 3 5 7 8 10 11 Faculty of Medicine, Suez University, Suez, Egypt, Suez, As Suways, Egypt 2Faculty of Oral and Dental Medicine, Egyptian Russian University, Badr City, Al Qahirah, Egypt 3Faculty of Medicine, Suez University, Suez, As Suways, Egypt 4Faculty of Medicine, Hashemite University, Zarqa, Jordan, Zarqa, Az Zarqa’, Jordan 5Faculty of Medicine, Jordan University of Science and Technology, Irbid, Jordan, Irbid, Irbid, Jordan 6Faculty of Medicine, Beni Suef University, Beni Suef, Egypt, Bani Suwayf, Bani Suwayf, Egypt 7Faculty of Medicine, Yarmouk University, Irbid, Jordan, Irbid, Irbid, Jordan 8Faculty of Medicine, University of Khartoum, Khartoum, Sudan, Khartoum, Khartoum, Sudan 9Faculty of Medicine, Tanta University, Tanta, Egypt, Tanta, Al Gharbiyah, Egypt 10Faculty of Medicine, Al-Azhar University, Damietta, Egypt, Damietta, Dumyat, Egypt 11Faculty of Medicine, Sohag University, Sohag, Egypt, Sohag, Suhaj, Egypt Forest Plot: Serious Adverse Events from Oral Antivirals (FAERS 2020–2023) This forest plot presents Reporting Odds Ratios (RORs) and 95% confidence intervals for serious adverse events linked to oral antivirals. Nirmatrelvir-ritonavir showed the strongest signals for drug–drug interactions (ROR: 4.83) and hepatic injury (ROR: 2.89). Molnupiravir was associated with neurological events and AKI. These findings highlight real-world safety patterns that inform risk-benefit assessment during antiviral therapy. Methods. A retrospective analysis of FAERS data from January 2020 to December 2023 was conducted. Reports involving favipiravir, molnupiravir, and nirmatrelvir-ritonavir were extracted. SAEs were defined per FDA criteria (death, lifethreatening event, hospitalization, disability). Event categories included hepatic injury, acute kidney injury (AKI), cardiovascular events, hypersensitivity, and drug–drug interactions. Disproportionality was assessed using Reporting Odds Ratios (ROR) with 95% confidence intervals (CI). Annual report volume and severity trends were also analyzed. Results. A total of 11,547 SAE reports related to oral antivirals were included. Nirmatrelvir-ritonavir accounted for the majority (62.5%), with significant signals for drug–drug interactions (ROR: 4.83, 95% CI: 4.35–5.32) and hepatic injury (ROR: 2.89). Molnupiravir was associated with neurological symptoms (ROR: 2.14) and AKI (ROR: 1.76). Reports peaked in mid-2022 and declined with reduced community transmission and updated prescribing guidelines. Conclusion. This FAERS-based..
DOI record: { "DOI": "10.1093/ofid/ofaf695.1825", "ISSN": [ "2328-8957" ], "URL": "http://dx.doi.org/10.1093/ofid/ofaf695.1825", "abstract": "<jats:title>Abstract</jats:title>\n <jats:sec>\n <jats:title>Background</jats:title>\n <jats:p>The COVID-19 pandemic led to the widespread use of emergency-authorized and repurposed oral antivirals, including remdesivir (initial IV use, later oral analogues), favipiravir, molnupiravir, and nirmatrelvir-ritonavir (Paxlovid). While these agents have played a key role in outpatient COVID-19 management, their real-world safety profiles remain under continuous evaluation. This study aimed to assess the temporal trends and disproportionality of serious adverse events (SAEs) associated with oral antivirals during the pandemic using the U.S. FDA Adverse Event Reporting System (FAERS).Forest Plot: Serious Adverse Events from Oral Antivirals (FAERS 2020–2023)This forest plot presents Reporting Odds Ratios (RORs) and 95% confidence intervals for serious adverse events linked to oral antivirals. Nirmatrelvir-ritonavir showed the strongest signals for drug–drug interactions (ROR: 4.83) and hepatic injury (ROR: 2.89). Molnupiravir was associated with neurological events and AKI. These findings highlight real-world safety patterns that inform risk-benefit assessment during antiviral therapy.</jats:p>\n </jats:sec>\n <jats:sec>\n <jats:title>Methods</jats:title>\n <jats:p>A retrospective analysis of FAERS data from January 2020 to December 2023 was conducted. Reports involving favipiravir, molnupiravir, and nirmatrelvir-ritonavir were extracted. SAEs were defined per FDA criteria (death, life-threatening event, hospitalization, disability). Event categories included hepatic injury, acute kidney injury (AKI), cardiovascular events, hypersensitivity, and drug–drug interactions. Disproportionality was assessed using Reporting Odds Ratios (ROR) with 95% confidence intervals (CI). Annual report volume and severity trends were also analyzed.</jats:p>\n </jats:sec>\n <jats:sec>\n <jats:title>Results</jats:title>\n <jats:p>A total of 11,547 SAE reports related to oral antivirals were included. Nirmatrelvir-ritonavir accounted for the majority (62.5%), with significant signals for drug–drug interactions (ROR: 4.83, 95% CI: 4.35–5.32) and hepatic injury (ROR: 2.89). Molnupiravir was associated with neurological symptoms (ROR: 2.14) and AKI (ROR: 1.76). Reports peaked in mid-2022 and declined with reduced community transmission and updated prescribing guidelines.</jats:p>\n </jats:sec>\n <jats:sec>\n <jats:title>Conclusion</jats:title>\n <jats:p>This FAERS-based analysis highlights evolving safety trends of oral antivirals during the COVID-19 pandemic. Nirmatrelvir-ritonavir demonstrated notable risks for hepatotoxicity and interaction-related events, emphasizing the importance of medication reconciliation and patient monitoring. Real-time pharmacovigilance remains critical for safe deployment of emerging antivirals in outpatient care.</jats:p>\n </jats:sec>\n <jats:sec>\n <jats:title>Disclosures</jats:title>\n <jats:p>All Authors: No reported disclosures</jats:p>\n </jats:sec>", "article-number": "ofaf695.1825", "author": [ { "affiliation": [ { "name": "Durdans Hospital , Colombo, Western Province ,", "place": [ "Sri Lanka" ] } ], "family": "Siby", "given": "Ashin", "sequence": "first" }, { "affiliation": [ { "name": "Durdans Hospital , Colombo, Western Province ,", "place": [ "Sri Lanka" ] } ], "family": "Mathew", "given": "Manu", "sequence": "additional" }, { "affiliation": [ { "name": "Durdans Hospital , Colombo, Western Province ,", "place": [ "Sri Lanka" ] } ], "family": "John", "given": "Jose T", "sequence": "additional" } ], "container-title": "Open Forum Infectious Diseases", "content-domain": { "crossmark-restriction": false, "domain": [] }, "created": { "date-parts": [ [ 2026, 1, 12 ] ], "date-time": "2026-01-12T07:29:47Z", "timestamp": 1768202987000 }, "deposited": { "date-parts": [ [ 2026, 1, 12 ] ], "date-time": "2026-01-12T07:41:46Z", "timestamp": 1768203706000 }, "indexed": { "date-parts": [ [ 2026, 1, 12 ] ], "date-time": "2026-01-12T10:39:42Z", "timestamp": 1768214382770, "version": "3.49.0" }, "is-referenced-by-count": 0, "issue": "Supplement_1", "issued": { "date-parts": [ [ 2026, 1 ] ] }, "journal-issue": { "issue": "Supplement_1", "published-print": { "date-parts": [ [ 2026, 1, 11 ] ] } }, "language": "en", "license": [ { "URL": "https://creativecommons.org/licenses/by/4.0/", "content-version": "vor", "delay-in-days": 11, "start": { "date-parts": [ [ 2026, 1, 12 ] ], "date-time": "2026-01-12T00:00:00Z", "timestamp": 1768176000000 } } ], "link": [ { "URL": "https://academic.oup.com/ofid/article-pdf/13/Supplement_1/ofaf695.1825/66354930/ofaf695.1825.pdf", "content-type": "application/pdf", "content-version": "vor", "intended-application": "syndication" }, { "URL": "https://academic.oup.com/ofid/article-pdf/13/Supplement_1/ofaf695.1825/66354930/ofaf695.1825.pdf", "content-type": "unspecified", "content-version": "vor", "intended-application": "similarity-checking" } ], "member": "286", "original-title": [], "prefix": "10.1093", "published": { "date-parts": [ [ 2026, 1 ] ] }, "published-online": { "date-parts": [ [ 2026, 1, 11 ] ] }, "published-other": { "date-parts": [ [ 2026, 1 ] ] }, "published-print": { "date-parts": [ [ 2026, 1, 11 ] ] }, "publisher": "Oxford University Press (OUP)", "reference-count": 0, "references-count": 0, "relation": {}, "resource": { "primary": { "URL": "https://academic.oup.com/ofid/article/doi/10.1093/ofid/ofaf695.1825/8422023" } }, "score": 1, "short-title": [], "source": "Crossref", "subject": [], "subtitle": [], "title": "P-1650. Temporal Trends in Serious Adverse Events Associated with Oral Antivirals During the COVID-19 Pandemic: Insights from the FAERS Database (2020–2023)", "type": "journal-article", "volume": "13" }
Please send us corrections, updates, or comments. c19early involves the extraction of 200,000+ datapoints from thousands of papers. Community updates help ensure high accuracy. Treatments and other interventions are complementary. All practical, effective, and safe means should be used based on risk/benefit analysis. No treatment or intervention is 100% available and effective for all current and future variants. We do not provide medical advice. Before taking any medication, consult a qualified physician who can provide personalized advice and details of risks and benefits based on your medical history and situation. IMA and WCH provide treatment protocols.
  or use drag and drop   
Submit