IL-1β and TNF drive endothelial dysfunction and coagulopathy in acute COVID-19

Mostafavi et al., bioRxiv, doi:10.64898/2026.03.21.713333, Mar 2026
In vitro and mouse study showing benefit with dexamethasone, adalimumab (anti-TNF), anakinra (IL-1R antagonist), and anti-IL-1β antibodies in preventing SARS-CoV-2-induced endothelial dysfunction and coagulopathy.
Mostafavi et al., 25 Mar 2026, Australia, preprint, 13 authors. Contact: l.labzin@uq.edu.au.
In vitro studies are an important part of preclinical research, however results may be very different in vivo.
Abstract: bioRxiv preprint doi: https://doi.org/10.64898/2026.03.21.713333; this version posted March 25, 2026. The copyright holder for this preprint (which was not certified by peer review) is the author/funder. All rights reserved. No reuse allowed without permission. 1 IL-1β and TNF drive endothelial dysfunction and coagulopathy in acute COVID-19. 2 3 Helen Mostafavi1, Brittany Hill1,2, Christina Nalkurthi2, Stefanie M Bader3,4, Yanshan Zhu1,, 4 Alexander Yu1, Philip M. Hansbro2, Marcel Doerflinger3,4, Matt D. Johansen2, Kirsty R. 5 Short5,6, Keng Yih Chew5,*, Emma J Gordon1,*, Larisa I Labzin1,6,7* 6 7 1 8 4072, Australia. 9 2 Institute for Molecular Bioscience (IMB), The University of Queensland, Brisbane, QLD Centre for Inflammation, Centenary Institute and University of Technology Sydney, Faculty 10 of Science, Sydney, NSW, Australia 11 3 12 Australia. 13 4 Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia 14 5 School of Chemistry and Molecular Biosciences, The University of Queensland, Brisbane, 15 QLD 4072, Australia. 16 6 17 QLD 4072, Australia 18 7 19 Behavioural Sciences, The University of Queensland, Brisbane, Australia. The Walter and Eliza Hall Institute of Medical Research (WEHI), Parkville, VIC 3052, Australian Infectious Diseases Research Centre, The University of Queensland, Brisbane, Centre for Cardiovascular Health and Research, Faculty of Health, Medicine and 20 21 * 22 Corresponding author. Email: l.labzin@uq.edu.au 23 These authors contributed equally. bioRxiv preprint doi: https://doi.org/10.64898/2026.03.21.713333; this version posted March 25, 2026. The copyright holder for this preprint (which was not certified by peer review) is the author/funder. All rights reserved. No reuse allowed without permission. 24 Abstract 25 26 Vascular dysfunction and coagulopathy are hallmarks of severe COVID-19. How SARS- 27 CoV-2 infection drives endothelial dysfunction, despite the virus not infecting or replicating 28 in endothelial cells, remains controversial. Here, we used an in vitro co-culture model of the 29 human pulmonary epithelial-endothelial cell barrier to investigate which inflammatory 30 mediators drive endothelial dysfunction during SARS-CoV-2 infection. SARS-CoV-2 31 infection of primary human bronchial epithelial cells increased adjacent endothelial cell 32 expression of the leukocyte adhesion marker ICAM-1, disrupted endothelial VE-cadherin 33 junctions, promoted endothelial cell death, and promoted platelet adherence to gaps in the 34 endothelial monolayers. Dexamethasone treatment rescued these dysregulated endothelial 35 phenotypes in infected co-cultures, confirming that inflammatory signalling was the primary 36 driver of SARS-CoV-2-induced endothelial dysfunction. Specifically, epithelial-derived TNF 37 and IL-1β promoted endothelial dysfunction, as inhibition of TNF or IL-1R signalling 38 blocked SARS-CoV-2-induced endothelial dysfunction in co-cultures. SARS-CoV-2-infected 39 wild-type mice, but not TNF, IL-1β, or TNF/IL-1β− deficient mice, displayed increased 40 endothelial ICAM-1 expression, while an anti-IL-1β monoclonal antibody prevented SARS- 41 CoV-2-induced ICAM-1 expression and fibrin deposition in aged K18-ACE2 mice. Our data 42 indicate that TNF and IL-1β are the specific cytokines that drive multiple aspects of 43 endothelial dysfunction during acute SARS-CoV-2 infection, and that..
DOI record: { "DOI": "10.64898/2026.03.21.713333", "URL": "http://dx.doi.org/10.64898/2026.03.21.713333", "abstract": "<jats:title>Abstract</jats:title>\n <jats:p>\n Vascular dysfunction and coagulopathy are hallmarks of severe COVID-19. How SARS-CoV-2 infection drives endothelial dysfunction, despite the virus not infecting or replicating in endothelial cells, remains controversial. Here, we used an\n <jats:italic>in vitro</jats:italic>\n co-culture model of the human pulmonary epithelial-endothelial cell barrier to investigate which inflammatory mediators drive endothelial dysfunction during SARS-CoV-2 infection. SARS-CoV-2 infection of primary human bronchial epithelial cells increased adjacent endothelial cell expression of the leukocyte adhesion marker ICAM-1, disrupted endothelial VE-cadherin junctions, promoted endothelial cell death, and promoted platelet adherence to gaps in the endothelial monolayers. Dexamethasone treatment rescued these dysregulated endothelial phenotypes in infected co-cultures, confirming that inflammatory signalling was the primary driver of SARS-CoV-2-induced endothelial dysfunction. Specifically, epithelial-derived TNF and IL-1β promoted endothelial dysfunction, as inhibition of TNF or IL-1R signalling blocked SARS-CoV-2-induced endothelial dysfunction in co-cultures. SARS-CoV-2-infected wild-type mice, but not TNF, IL-1β, or TNF/IL-1β− deficient mice, displayed increased endothelial ICAM-1 expression, while an anti-IL-1β monoclonal antibody prevented SARS-CoV-2-induced ICAM-1 expression and fibrin deposition in aged K18-ACE2 mice. Our data indicate that TNF and IL-1β are the specific cytokines that drive multiple aspects of endothelial dysfunction during acute SARS-CoV-2 infection, and that inhibiting their signalling pathways may provide therapeutic benefit in preventing vascular complications of COVID-19.\n </jats:p>", "accepted": { "date-parts": [ [ 2026, 3, 25 ] ] }, "author": [ { "affiliation": [ { "name": "Institute for Molecular Bioscience (IMB), The University of Queensland, Brisbane, QLD 4072, Australia" } ], "family": "Mostafavi", "given": "Helen", "sequence": "first" }, { "affiliation": [ { "name": "Institute for Molecular Bioscience (IMB), The University of Queensland, Brisbane, QLD 4072, Australia" }, { "name": "Centre for Inflammation, Centenary Institute and University of Technology Sydney, Faculty of Science, Sydney, NSW, Australia" } ], "family": "Hill", "given": "Brittany", "sequence": "additional" }, { "affiliation": [ { "name": "Centre for Inflammation, Centenary Institute and University of Technology Sydney, Faculty of Science, Sydney, NSW, Australia" } ], "family": "Nalkurthi", "given": "Christina", "sequence": "additional" }, { "affiliation": [ { "name": "The Walter and Eliza Hall Institute of Medical Research (WEHI), Parkville, VIC 3052, Australia" }, { "name": "Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia" } ], "family": "Bader", "given": "Stefanie M", "sequence": "additional" }, { "affiliation": [ { "name": "Institute for Molecular Bioscience (IMB), The University of Queensland, Brisbane, QLD 4072, Australia" } ], "family": "Zhu", "given": "Yanshan", "sequence": "additional" }, { "affiliation": [ { "name": "Institute for Molecular Bioscience (IMB), The University of Queensland, Brisbane, QLD 4072, Australia" } ], "family": "Yu", "given": "Alexander", "sequence": "additional" }, { "affiliation": [ { "name": "Centre for Inflammation, Centenary Institute and University of Technology Sydney, Faculty of Science, Sydney, NSW, Australia" } ], "family": "Hansbro", "given": "Philip M.", "sequence": "additional" }, { "affiliation": [ { "name": "The Walter and Eliza Hall Institute of Medical Research (WEHI), Parkville, VIC 3052, Australia" }, { "name": "Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia" } ], "family": "Doerflinger", "given": "Marcel", "sequence": "additional" }, { "affiliation": [ { "name": "Centre for Inflammation, Centenary Institute and University of Technology Sydney, Faculty of Science, Sydney, NSW, Australia" } ], "family": "Johansen", "given": "Matt D.", "sequence": "additional" }, { "affiliation": [ { "name": "School of Chemistry and Molecular Biosciences, The University of Queensland, Brisbane, QLD 4072, Australia" }, { "name": "Australian Infectious Diseases Research Centre, The University of Queensland, Brisbane, QLD 4072, Australia" } ], "family": "Short", "given": "Kirsty R.", "sequence": "additional" }, { "affiliation": [ { "name": "School of 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